At NINGBO INNO PHARMCHEM CO.,LTD., we are dedicated to providing high-quality pharmaceutical ingredients. Today, we focus on Phenprobamate, a compound with a significant history and ongoing relevance in therapeutic applications. Understanding its properties is key for researchers and formulators aiming to develop effective treatments.

Phenprobamate is a centrally acting skeletal muscle relaxant that also possesses notable sedative and anticonvulsant properties. This multifaceted profile has led to its use in various clinical settings. Historically, it served as an anxiolytic and is still recognized for its utility in managing muscle cramps and spasticity. While newer medications have emerged, Phenprobamate remains a subject of interest due to its established pharmacological actions.

The core of Phenprobamate's efficacy lies in its mechanism of action, which is believed to heavily involve the potentiation of gamma-aminobutyric acid (GABA) neurotransmission. GABA is the primary inhibitory neurotransmitter in the central nervous system, and by enhancing its effects, Phenprobamate helps to reduce neuronal excitability. This reduction in excitability is what allows it to effectively alleviate muscle spasms and exert its anxiolytic and sedative effects. The precise dosage can vary, with common recommendations ranging from 400 to 800 mg, up to three times daily, though consultation with healthcare professionals is paramount.

The metabolism of Phenprobamate involves oxidative degradation of its carbamate group and ortho-hydroxylation of the benzene ring, with elimination occurring primarily through the kidneys. This pharmacokinetic profile is essential for understanding its duration of action and potential drug interactions. NINGBO INNO PHARMCHEM CO.,LTD. ensures that the Phenprobamate we supply adheres to strict quality standards, crucial for consistent therapeutic outcomes.

While Phenprobamate has been used for decades, it's important for formulators to be aware of its profile. When considering the purchase of Phenprobamate, partners often inquire about the best price and reliable sourcing for pharmaceutical intermediates. NINGBO INNO PHARMCHEM CO.,LTD. stands as a trusted supplier, committed to providing competitive pricing and consistent availability for Phenprobamate to support your research and development needs. We understand the critical role that high-purity Phenprobamate plays in creating effective pharmaceutical products for muscle relaxation and anxiety relief.