Exploring Tofisopam (CAS 22345-47-7): An Atypical Benzodiazepine Derivative
Uncover the chemical properties, therapeutic uses, and pharmacological insights of this unique 2,3-benzodiazepine compound.
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Tofisopam
Tofisopam, identified by its CAS number 22345-47-7, is a distinct 2,3-benzodiazepine derivative with a unique pharmacological profile. Unlike conventional benzodiazepines, it lacks significant anticonvulsant, sedative, and muscle relaxant properties, positioning it as an atypical anxiolytic. Its primary mechanism involves modulating GABAA receptors, contributing to its therapeutic effects in managing anxiety and depression. Understanding the Tofisopam GABAergic mechanism is crucial for its application in treating mood disorders.
- Detailed insights into Tofisopam chemical properties are essential for research and development, covering its molecular formula C22H26N2O4 and molecular weight of 382.45.
- Exploring the Tofisopam applications reveals its use in treating depression and associated anxiety, offering a novel approach to mental health support.
- The Tofisopam synthesis pathways are of interest to chemical manufacturers aiming for efficient production of this pharmaceutical intermediate.
- Researching the Tofisopam safety information is paramount, especially its classification as a Category D pregnancy drug and its potential for habit formation.
Key Advantages of Tofisopam
Unique Anxiolytic Profile
Tofisopam offers a distinct anxiolytic action without the typical sedative or muscle relaxant side effects associated with other benzodiazepines, making it suitable for daytime use.
Broad Therapeutic Potential
Beyond anxiety, studies suggest Tofisopam's potential in treating depression and even the negative symptoms of psychosis, expanding its therapeutic scope.
GABA Receptor Modulation
Understanding the Tofisopam GABAergic mechanism provides a foundation for developing more targeted treatments for neurological and psychological conditions.
Key Applications
Anxiety Treatment
As a key application, Tofisopam is prescribed to manage various anxiety disorders, providing relief from excessive fear and worry.
Depression Management
The drug plays a vital role in treating depression and related anxiety, improving mood and overall quality of life for patients.
Pharmaceutical Intermediate
Its chemical structure makes Tofisopam a valuable intermediate in the synthesis of other complex pharmaceutical compounds and research chemicals.
Neuroscience Research
Researchers utilize Tofisopam to study the intricacies of GABAergic neurotransmission and benzodiazepine receptor binding for a deeper understanding of brain function.
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