The Role of 2-Iodobenzotrifluoride in Modern Organic Synthesis
In the intricate world of organic synthesis, the availability of versatile and reactive intermediates is the cornerstone of innovation. 2-Iodobenzotrifluoride (CAS 444-29-1) has firmly established itself as such a compound, offering chemists a powerful tool for constructing complex molecular architectures. Its utility spans across various synthetic strategies, but it is particularly prized for its role in modern cross-coupling reactions.
The molecular structure of 2-Iodobenzotrifluoride, featuring a carbon-iodine bond and a trifluoromethyl substituent on an aromatic ring, is the source of its synthetic prowess. The carbon-iodine bond is relatively weak and readily undergoes oxidative addition with transition metal catalysts, a key step in many palladium-catalyzed cross-coupling reactions like Suzuki, Heck, Sonogashira, and Stille couplings. These reactions are indispensable for forming new carbon-carbon bonds, enabling the assembly of diverse organic frameworks. Researchers actively seeking to buy 2-Iodobenzotrifluoride often do so to leverage these powerful synthetic methodologies.
The presence of the trifluoromethyl (CF3) group is another significant advantage. This electron-withdrawing substituent can influence the reactivity of the aromatic ring and the overall properties of the final molecule. In pharmaceuticals and agrochemicals, the incorporation of CF3 groups is a common strategy to enhance biological activity, metabolic stability, and bioavailability. Consequently, 2-Iodobenzotrifluoride serves as an efficient way to introduce both an iodine handle for coupling and a trifluoromethyl group into target molecules simultaneously.
As a leading manufacturer and supplier of fine chemicals, NINGBO INNO PHARMCHEM CO.,LTD. provides high-quality 2-Iodobenzotrifluoride to support your synthetic chemistry needs. Our commitment to stringent quality control ensures product purity, which is vital for achieving reproducible and high-yielding reactions. For procurement managers and research scientists, sourcing this key intermediate from a reliable manufacturer in China offers cost-effectiveness and assured supply. We encourage you to inquire about pricing and availability for your next synthetic project.
Perspectives & Insights
Molecule Vision 7
“This electron-withdrawing substituent can influence the reactivity of the aromatic ring and the overall properties of the final molecule.”
Alpha Origin 24
“In pharmaceuticals and agrochemicals, the incorporation of CF3 groups is a common strategy to enhance biological activity, metabolic stability, and bioavailability.”
Future Analyst X
“Consequently, 2-Iodobenzotrifluoride serves as an efficient way to introduce both an iodine handle for coupling and a trifluoromethyl group into target molecules simultaneously.”