Intermediates

1-Iodo-4,4,4-trifluorobutane

  • CAS No.461-17-6
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 1-iodo-4,4,4-trifluorobutane (CAS 461-17-6) is a versatile fluorinated building block widely used as an intermediate in advanced organic synthesis for pharmaceuticals, agrochemicals, and novel materials.

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Product Technical Details

Product Overview

1-Iodo-4,4,4-trifluorobutane (CAS 461-17-6) is a high-value fluorinated alkyl halide employed extensively as a synthetic intermediate in modern organic chemistry. With its unique combination of a reactive iodine atom and a strongly electron-withdrawing trifluoromethyl group, this compound serves as a key building block for constructing complex fluorinated molecules essential in pharmaceutical R&D, agrochemical innovation, and advanced material science.

Specifications

Molecular FormulaC₄H₆F₃I
Molecular Weight237.99 g/mol
AppearanceClear liquid
Assay (GC)≥98.0%
Moisture≤0.1%
Density1.85 g/cm³
Boiling Point126°C
Flash Point>100°C
Refractive Index1.4326

Industrial Applications

This fluorinated intermediate plays a critical role in multi-step syntheses where controlled introduction of a -CF₃-containing alkyl chain is required. Its primary applications include:

  • Serving as a precursor in the preparation of fluorinated heterocycles and bioactive compounds during early-stage drug discovery.
  • Facilitating cross-coupling reactions (e.g., Suzuki, Negishi) to construct C–C bonds in fluorinated scaffolds.
  • Acting as an alkylating agent in the development of novel agrochemicals with enhanced metabolic stability.
  • Supporting the synthesis of specialty monomers for high-performance fluoropolymers.

Manufactured under stringent quality control protocols, our 1-iodo-4,4,4-trifluorobutane meets international standards for industrial-scale use. It is typically packed in 200 kg drums and should be stored in a cool, well-ventilated area away from light and moisture to maintain stability and reactivity.