Intermediates

(2R,3S)-3-Phenylisoserine

  • CAS No.136561-53-0
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity (2R,3S)-3-Phenylisoserine, a key chiral intermediate for the synthesis of Cabazitaxel and other advanced oncology APIs.

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Product Technical Details

Product Overview

(2R,3S)-3-Phenylisoserine is a high-value chiral amino acid derivative widely employed as a critical building block in the pharmaceutical industry. With its defined stereochemistry and functional group array, it serves as an essential intermediate in the synthesis of complex taxane-based therapeutics, most notably Cabazitaxel (CAS: 183133-96-2), a second-generation microtubule inhibitor used in oncology treatments.

Specifications

Molecular FormulaC9H11NO3
Molecular Weight167.205 g/mol
Density1.2 ± 0.1 g/cm³
Boiling Point360.6 ± 37.0 °C at 760 mmHg
Flash Point171.9 ± 26.5 °C
Vapour Pressure0.0 ± 0.8 mmHg at 25°C
Refractive Index1.594
Assay≥98.0%
AppearanceWhite to off-white powder

Industrial Applications

This compound is exclusively utilized as a synthetic intermediate in regulated pharmaceutical manufacturing environments. Its primary application lies in the stereoselective construction of the side chain of Cabazitaxel, where precise chirality at the 2R,3S positions is crucial for biological activity and regulatory compliance. Due to its role in enabling complex active pharmaceutical ingredients (APIs), (2R,3S)-3-Phenylisoserine is produced under stringent quality control protocols aligned with ICH guidelines.

  • Enables high-yield, stereospecific coupling in taxane derivatization
  • Supplied with full analytical documentation including COA and HPLC chromatograms
  • Compatible with GMP-compliant manufacturing workflows
  • Stable under recommended storage conditions for extended shelf life

For industrial-scale procurement, the product is typically packed in 25 kg fiber drums with double-layer polyethylene liners, though custom packaging solutions are available upon request. Storage should be in a cool, dry, and well-ventilated area away from incompatible materials.