Intermediates

3,6-Dichloropyridazine

  • CAS No.141-30-0
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 3,6-Dichloropyridazine (CAS 141-30-0), a key building block for pharmaceutical intermediates such as Sulfachloropyridazine.

Request Bulk Pricing

Product Technical Details

Product Overview

3,6-Dichloropyridazine (CAS 141-30-0) is a high-value heterocyclic compound widely employed as a critical intermediate in the synthesis of active pharmaceutical ingredients (APIs). Its rigid diazine core substituted with two chlorine atoms at positions 3 and 6 offers excellent reactivity for nucleophilic aromatic substitution, enabling efficient derivatization in multi-step syntheses. This compound serves as a foundational scaffold in the production of sulfonamide-based therapeutics, including Sulfachloropyridazine (CAS 80-32-0).

Specifications

Molecular FormulaC4H2Cl2N2
Molecular Weight148.98 g/mol
Melting Point65–69 °C (lit.)
Boiling Point277.0 ± 20.0 °C at 760 mmHg
Density1.5 ± 0.1 g/cm³
LogP0.90
AppearanceWhite or off-white crystalline solid
Assay≥99.0%
Loss on Drying (IR-lamp)≤0.1%
Water Content (K.F.)≤0.1%

Industrial Applications

As a versatile synthetic intermediate, 3,6-Dichloropyridazine is primarily utilized in the pharmaceutical industry for constructing complex molecular architectures. Its applications include:

  • Serving as a precursor in the manufacture of sulfonamide antibiotics like Sulfachloropyridazine.
  • Enabling the development of novel neurological and anti-infective therapeutics through regioselective functionalization.
  • Supporting advanced organic synthesis campaigns requiring halogenated diazine motifs.

Due to its sensitivity to moisture and thermal degradation, it must be stored in a cool, dry, and well-ventilated environment with the container tightly sealed. Standard packaging is 25 kg per drum, with custom configurations available upon request.