Intermediates

3-Amino-2-fluoropyridine

  • CAS No.1597-33-7
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 3-Amino-2-fluoropyridine (CAS 1597-33-7), a key fluorinated heterocyclic intermediate for pharmaceutical R&D and API synthesis.

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Product Technical Details

Product Overview

3-Amino-2-fluoropyridine (CAS 1597-33-7) is a high-value fluorinated heterocyclic compound widely employed as a critical building block in the synthesis of advanced pharmaceutical intermediates. With its unique combination of an amino group and a fluorine atom on the pyridine ring, it offers versatile reactivity for cross-coupling, nucleophilic substitution, and cyclization reactions, making it indispensable in modern medicinal chemistry workflows.

Specifications

Molecular FormulaC5H5FN2
Molecular Weight112.11 g/mol
AppearanceYellow liquid
Purity≥99.0%
Density1.3 ± 0.1 g/cm³
Boiling Point243.2 ± 20.0 °C at 760 mmHg
Flash Point100.9 ± 21.8 °C
Refractive Index1.554
Packaging25 kg/drum
StorageStore in a tightly closed container in a cool, dry place

Industrial Applications

As a specialized fluoro-heterocyclic intermediate, 3-Amino-2-fluoropyridine serves as a foundational scaffold in the development of complex pharmaceutical APIs, particularly in neurological therapeutics and targeted kinase inhibitors. Its strategic placement of fluorine enhances metabolic stability and bioavailability in drug candidates.

  • Ideal for Suzuki, Buchwald-Hartwig, and other Pd-catalyzed transformations
  • Enables rapid diversification of molecular libraries in early-stage drug discovery
  • Consistent batch-to-batch quality ensures reliable performance in GMP-compliant synthesis
  • Sourced from ISO-certified manufacturing facilities with full traceability