Intermediates

3-Bromo-2-methoxypyridine

  • CAS No.13472-59-8
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 3-Bromo-2-methoxypyridine (CAS 13472-59-8), a versatile pyridine-based intermediate for advanced organic synthesis in pharmaceutical and agrochemical manufacturing.

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Product Technical Details

Product Overview

3-Bromo-2-methoxypyridine is a high-value halogenated heterocyclic compound widely employed as a key building block in modern organic synthesis. With its reactive bromine atom adjacent to an electron-donating methoxy group on the pyridine ring, this molecule offers exceptional regioselectivity for cross-coupling reactions such as Suzuki, Stille, and Negishi protocols. It serves as a critical intermediate in the development of active pharmaceutical ingredients (APIs), crop protection agents, and functional materials.

Specifications

Molecular FormulaC6H6BrNO
Molecular Weight188.02 g/mol
CAS Number13472-59-8
AppearanceColorless liquid
Purity≥99.0%
Density1.5856 g/cm³
Boiling Point190.4°C
Flash Point93°C
Refractive Index1.566

Industrial Applications

As a specialized pyridine derivative, 3-Bromo-2-methoxypyridine is primarily utilized in the pharmaceutical and agrochemical sectors for constructing complex molecular architectures. Its structural features enable efficient functionalization at the C3 position, facilitating the introduction of aryl, alkyl, or heteroaryl moieties. This intermediate supports the scalable synthesis of drug candidates targeting neurological, oncological, and metabolic disorders, as well as next-generation herbicides and insecticides.

  • Enables precise C–C and C–N bond formation via transition-metal catalysis
  • Compatible with standard handling protocols for moisture-sensitive reagents
  • Supplied in industrial-grade packaging with full analytical documentation (COA)

Stored in a cool, well-ventilated area away from ignition sources, this product maintains stability under recommended conditions and is available in 200 kg drums or custom packaging upon request.