Intermediates

3-Bromo-4-fluorophenol

  • CAS No.27407-11-0
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 3-Bromo-4-fluorophenol (CAS 27407-11-0), a versatile halogenated aromatic intermediate for advanced organic synthesis in pharmaceutical and agrochemical R&D.

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Product Technical Details

Product Overview

3-Bromo-4-fluorophenol is a high-value halogenated aromatic compound widely employed as a key building block in the synthesis of complex organic molecules. With its dual functionality—featuring both bromo and fluoro substituents on the phenolic ring—it offers excellent regioselectivity for cross-coupling reactions, nucleophilic aromatic substitutions, and directed ortho-metalation strategies. This intermediate is particularly valuable in the development of active pharmaceutical ingredients (APIs) and specialty agrochemicals where precise molecular architecture is critical.

Specifications

Molecular FormulaC6H4BrFO
Molecular Weight190.998 g/mol
CAS Number27407-11-0
AppearanceYellow oil
Assay≥98.0%
Density1.8 ± 0.1 g/cm³
Boiling Point240.5 ± 20.0 °C at 760 mmHg
Flash Point99.2 ± 21.8 °C
Vapour Pressure0.0 ± 0.5 mmHg at 25°C
Refractive Index1.576

Industrial Applications

As a specialized intermediate, 3-Bromo-4-fluorophenol serves as a strategic precursor in multi-step synthetic pathways. Its applications include:

  • Construction of biaryl scaffolds via Suzuki-Miyaura or Ullmann couplings
  • Synthesis of fluorinated phenolic derivatives for medicinal chemistry programs
  • Development of novel ligands and functional materials in materials science
  • Preparation of herbicidal and fungicidal agents in crop protection chemistry

Due to its reactivity profile and stability under standard handling conditions, it is well-suited for scale-up in GMP-compliant manufacturing environments. The compound should be stored in a cool, dry, and well-ventilated area away from oxidizing agents and strong bases to maintain integrity and performance.