Intermediates

3-Fluoro-4-(trifluoromethoxy)aniline

  • CAS No.1017779-69-9
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 3-Fluoro-4-(trifluoromethoxy)aniline (CAS 1017779-69-9), a key fluorinated intermediate for advanced organic synthesis in pharmaceutical and agrochemical R&D.

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Product Technical Details

Product Overview

3-Fluoro-4-(trifluoromethoxy)aniline is a high-value fluorinated aromatic amine widely employed as a critical building block in the synthesis of complex organic molecules. With its unique combination of electron-withdrawing trifluoromethoxy and fluoro substituents, this compound offers enhanced metabolic stability and lipophilicity—properties highly sought after in modern medicinal chemistry and crop protection agent development.

Specifications

Molecular FormulaC₇H₅F₄NO
Molecular Weight195.11 g/mol
AppearanceColourless to yellow to light brown liquid
Purity (GC)≥99.0%
StorageStore in a cool, well-ventilated area away from heat and incompatible materials
Packaging200 kg/drum; custom packaging available upon request

Industrial Applications

As a specialized fluoroaromatic intermediate, 3-Fluoro-4-(trifluoromethoxy)aniline serves primarily in the early- to mid-stage synthesis of active pharmaceutical ingredients (APIs) and agrochemical actives. Its structural motif enables efficient derivatization via diazotization, acylation, or cross-coupling reactions, facilitating rapid scaffold diversification in drug discovery pipelines.

  • Ideal for constructing novel heterocyclic systems with improved pharmacokinetic profiles
  • Used in the development of selective enzyme inhibitors and receptor modulators
  • Supports green chemistry initiatives through high-yield, low-waste synthetic routes

Manufactured under stringent quality control protocols, our product meets global regulatory standards for use in GMP-compliant research and pilot-scale production environments.