Intermediates

4,7-Dichloroquinoline

  • CAS No.86-98-6
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 4,7-Dichloroquinoline (CAS 86-98-6), a key pharmaceutical intermediate for antimalarial and heterocyclic compound synthesis. Assay ≥99.0%, manufactured at 20-ton monthly capacity in China.

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Product Technical Details

Product Overview

4,7-Dichloroquinoline is a critical heterocyclic building block widely employed in the synthesis of advanced pharmaceutical intermediates, particularly in the development of antimalarial agents and other nitrogen-containing bioactive molecules. As a high-value quinoline derivative, it serves as a foundational scaffold in multi-step organic syntheses requiring regioselective functionalization.

Specifications

AppearanceLight yellow solid or light yellow crystalline solid
Melting Point83–87 °C
Assay (GC/HPLC)≥99.0%
Moisture (Karl Fischer)≤1.0%
4,5-Dichloroquinoline≤0.5%
7-Chloro-4-hydroxyquinoline≤0.3%
Other Single Impurities≤0.5%

Industrial Applications

This compound is primarily utilized as a synthetic intermediate in the pharmaceutical industry. Its dual chlorine substitution pattern enables selective nucleophilic aromatic substitution reactions, facilitating the construction of complex molecular architectures. Key application areas include:

  • Synthesis of chloroquine-related antimalarial drug candidates
  • Preparation of kinase inhibitors and other targeted therapeutics
  • Building block for fluorescent probes and agrochemical research
  • Intermediate in the production of specialty ligands for catalysis

Manufactured under stringent quality control systems compliant with international GMP guidelines, our 4,7-Dichloroquinoline is produced at a scale of 20 metric tons per month, ensuring reliable supply for global API manufacturers and R&D institutions.