Intermediates

4-Amino-2,6-dimethoxypyrimidine

  • CAS No.3289-50-7
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 4-Amino-2,6-dimethoxypyrimidine (CAS 3289-50-7), a key pharmaceutical intermediate in the synthesis of sulfonamide antibiotics such as Sulphadimethoxine.

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Product Technical Details

Product Overview

4-Amino-2,6-dimethoxypyrimidine is a high-value heterocyclic organic compound widely employed as a critical building block in the pharmaceutical industry. With the CAS registry number 3289-50-7, this molecule serves as an essential intermediate in the synthesis of sulfonamide-class antimicrobial agents, particularly Sulphadimethoxine. Its well-defined reactivity and structural features make it indispensable for constructing complex pyrimidine-based active pharmaceutical ingredients (APIs).

Specifications

Molecular FormulaC6H9N3O2
Molecular Weight155.15 g/mol
EINECS Number221-946-2
Density1.2 ± 0.1 g/cm³
Boiling Point340.1 ± 45.0 °C at 760 mmHg
Melting Point149–152 °C (lit.)
Flash Point159.5 ± 28.7 °C
Refractive Index1.547
AppearanceWhite crystal
Assay≥95%
Residue on Ignition≤0.2%
Water Content≤0.5%

Industrial Applications

This compound is primarily utilized as a synthetic intermediate in the production of Sulphadimethoxine, a long-acting sulfonamide antibiotic used in veterinary and human medicine. Its role in facilitating selective functionalization of the pyrimidine core enables efficient, scalable routes to target APIs under GMP-compliant conditions.

  • Serves as a foundational scaffold for sulfonamide antibiotic synthesis
  • Compatible with standard amidation and nucleophilic substitution protocols
  • Supplied in industrial-grade purity suitable for multi-step pharmaceutical manufacturing

Handling and Storage

Store in a cool, well-ventilated warehouse away from heat sources and open flames. Maintain storage temperature below 37 °C. Packaging is typically provided in 25 kg drums, with custom options available upon request to meet specific logistical or regulatory requirements.