Intermediates

4-Methylsulfonylbenzaldehyde

  • CAS No.5398-77-6
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 4-Methylsulfonylbenzaldehyde (CAS 5398-77-6), a key pharmaceutical intermediate for the synthesis of chloramphenicol and thiamphenicol.

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Product Technical Details

Product Overview

4-Methylsulfonylbenzaldehyde (CAS 5398-77-6) is a high-value aromatic aldehyde widely employed as a critical building block in the synthesis of advanced pharmaceutical intermediates. This compound features a methylsulfonyl group at the para position of the benzaldehyde ring, imparting enhanced reactivity and stability for use in multi-step organic transformations.

Specifications

Molecular FormulaC8H8O3S
Molecular Weight184.21 g/mol
AppearanceLight yellow crystal powder
Purity≥99%
Moisture Content≤0.30%
Melting Point155–161 °C
Boiling Point378.3 °C at 760 mmHg
Density1.289 g/cm³
Flash Point242.1 °C
Refractive Index1.544

Industrial Applications

As a versatile synthetic intermediate, 4-Methylsulfonylbenzaldehyde serves as a foundational precursor in the production of several important antibiotics. It is primarily utilized in the manufacturing pathways of chloramphenicol (CAS 56-75-7) and thiamphenicol (CAS 15318-45-3), both of which are broad-spectrum antimicrobial agents used in human and veterinary medicine.

Key advantages of this intermediate include:

  • High chemical purity ensuring consistent reaction yields
  • Excellent thermal and oxidative stability during storage and processing
  • Compatibility with standard industrial-scale synthesis protocols
  • Reliable performance in nucleophilic addition and condensation reactions

Handling and Storage

Store in a cool, dry, and well-closed container away from moisture, strong light, and heat sources. Proper handling in accordance with local regulatory guidelines is recommended to maintain product integrity and ensure workplace safety.