Intermediates

6,7-Dimethoxy-4-hydroxyquinoline

  • CAS No.13425-93-9
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 6,7-Dimethoxy-4-hydroxyquinoline (CAS 13425-93-9), a key pharmaceutical intermediate for Tivozanib synthesis, manufactured to stringent quality standards.

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Product Technical Details

Product Overview

6,7-Dimethoxy-4-hydroxyquinoline is a high-value quinoline derivative widely employed as a critical building block in the synthesis of advanced pharmaceutical intermediates. With a molecular formula of C11H11NO3 and a molecular weight of 205.21 g/mol, this compound exhibits excellent reactivity and selectivity in heterocyclic chemistry, making it indispensable in modern medicinal chemistry workflows.

Specifications

AppearanceYellow to off-white crystalline powder
Purity (HPLC)≥98.0%
Loss on Drying≤1.0%
Residue on Ignition≤0.5%
Any Single Impurity≤0.5%
Total Impurities≤1.0%
Density1.206 g/cm³
Melting Point30°C
Boiling Point355.3°C
Flash Point168.7°C

Industrial Applications

This compound serves primarily as a specialized intermediate in the production of Tivozanib, a potent tyrosine kinase inhibitor used in oncology therapeutics. Its well-defined substitution pattern enables efficient regioselective functionalization during multi-step syntheses.

  • Enables streamlined access to complex quinoline-based active pharmaceutical ingredients (APIs)
  • Manufactured under strict GMP-aligned conditions to ensure batch-to-batch consistency
  • Suitable for scale-up in commercial pharmaceutical manufacturing environments

Packaging is typically provided in 25 kg drums, with custom options available upon request. The product should be stored in a cool, dry, and well-ventilated area, protected from moisture and direct sunlight. Please note that distribution may be restricted in jurisdictions where relevant patents are in force.