Intermediates

Boc-D-Tic-OH

  • CAS No.11592-35-1
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity Boc-D-Tic-OH (CAS 11592-35-1), a valuable chiral building block for pharmaceutical intermediates and complex organic synthesis.

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Product Technical Details

Product Overview

Boc-D-Tic-OH (N-tert-Butoxycarbonyl-D-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid) is a high-purity, non-natural amino acid derivative widely employed as a chiral intermediate in the synthesis of bioactive molecules and advanced pharmaceutical compounds. With a molecular formula of C15H19NO4 and a molecular weight of 277.32 g/mol, this compound features a rigid tetrahydroisoquinoline scaffold protected by a Boc group, offering excellent stability and stereoselectivity in multi-step syntheses.

Specifications

Molecular FormulaC15H19NO4
Molecular Weight277.32 g/mol
CAS Number11592-35-1
AppearanceWhite or Off-white Powder
Purity (HPLC)≥98%
Moisture Content<0.5%
Total Impurities<0.5%
Melting Point125–126°C
Density1.2 ± 0.1 g/cm³

Industrial Applications

Boc-D-Tic-OH serves primarily as a specialized intermediate in the development and large-scale manufacturing of complex pharmaceutical APIs, particularly those targeting neurological and cardiovascular therapeutic areas. Its constrained conformation and defined stereochemistry make it ideal for:

  • Peptidomimetic drug design and synthesis
  • Chiral auxiliary applications in asymmetric synthesis
  • Construction of protease inhibitors and receptor modulators
  • Advanced organic synthesis requiring enantiomerically pure scaffolds

As a non-controlled, non-hazardous fine chemical, it complies with international regulatory standards for research and commercial pharmaceutical production.

Handling and Storage

Store Boc-D-Tic-OH at 2–8°C in a tightly sealed container under dry, inert conditions. Protect from light, moisture, and prolonged exposure to ambient temperature to maintain integrity and purity. Standard industrial hygiene practices are recommended during handling.