Intermediates

Diethyl 2-acetamido-2-(2-phenylethyl)propanedioate

  • CAS No.5463-92-3
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity Diethyl 2-acetamido-2-(2-phenylethyl)propanedioate (CAS 5463-92-3) for pharmaceutical synthesis. Reliable bulk supply with ≥98% assay and full COA documentation.

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Product Technical Details

Product Overview

Diethyl 2-acetamido-2-(2-phenylethyl)propanedioate, commonly known as Diethyl 2-acetamido-2-phenethylmalonate, is a critical organic intermediate utilized extensively in the pharmaceutical industry. With the CAS registry number 5463-92-3, this compound serves as a key building block in the synthesis of complex therapeutic agents, most notably as a precursor in the manufacturing pathway of Fingolimod. Our facility specializes in the production of this high-value chemical, ensuring consistent quality and supply chain stability for global research and manufacturing partners.

As a specialized chemical manufacturer, we understand the stringent requirements of pharmaceutical synthesis. This compound features a stable malonate structure with an acetamido group, making it highly suitable for various organic transformation reactions. The molecular formula C17H23NO5 and molecular weight of 321.368 g/mol define its specific reactivity profile, which is essential for downstream processing in API production.

Technical Specifications

We adhere to strict quality control protocols to ensure every batch meets or exceeds industry standards. The following table outlines the key physical and chemical properties of our product:

ParameterSpecification
CAS Number5463-92-3
Molecular FormulaC17H23NO5
Molecular Weight321.368 g/mol
AppearanceWhite to light yellow powder
Assay (Purity)≥98.0%
Melting Point114-115°C
Density1.1±0.1 g/cm3
Boiling Point483.8±45.0°C at 760 mmHg
Flash Point246.4±28.7°C

Quality Assurance and Testing

Quality is the cornerstone of our manufacturing process. Each production lot undergoes rigorous analytical testing using advanced instrumentation such as High-Performance Liquid Chromatography (HPLC) and Nuclear Magnetic Resonance (NMR) spectroscopy. These tests verify the chemical identity, purity levels, and the absence of unwanted impurities. We provide a comprehensive Certificate of Analysis (COA) with every shipment, detailing the specific test results for that batch. This transparency allows our clients to maintain their own quality standards and regulatory compliance without interruption.

Industrial Applications

The primary application of Diethyl 2-acetamido-2-(2-phenylethyl)propanedioate is in the pharmaceutical sector, specifically as an intermediate for Fingolimod synthesis. Fingolimod is a significant medication used in the treatment of multiple sclerosis, and the precision of its intermediate components is vital for the efficacy and safety of the final drug product. Beyond this specific application, this chemical serves as a versatile reagent in organic synthesis laboratories for constructing complex molecular architectures involving phenethyl and malonate moieties. Its high purity ensures minimal side reactions during synthesis, optimizing yield and reducing waste.

Packaging, Storage, and Safety

To preserve the integrity of the chemical during transit and storage, we offer flexible packaging solutions. The standard packaging is 25 kg per drum, designed to protect the powder from moisture and physical damage. However, we accommodate custom packaging requirements based on client logistics and volume needs. For storage, the product should be kept in a cool, ventilated area away from direct sunlight and incompatible materials. Proper handling procedures, including the use of personal protective equipment (PPE), are recommended to ensure safety during industrial handling. Our global logistics network ensures timely delivery while maintaining the required storage conditions throughout the supply chain.