Intermediates

H-DL-Asp(OMe)-OMe Hydrochloride

  • CAS No.14358-33-9
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity H-DL-Asp(OMe)-OMe hydrochloride (CAS 14358-33-9), a key chiral building block for pharmaceutical intermediates and peptide synthesis.

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Product Technical Details

Product Overview

H-DL-Asp(OMe)-OMe hydrochloride is a protected derivative of aspartic acid, widely employed as a versatile intermediate in the synthesis of complex pharmaceutical APIs and bioactive peptides. With a molecular formula of C6H12ClNO4 and a molecular weight of 197.62 g/mol, this compound features dual methyl ester protection on the carboxylic acid groups, enhancing its stability and reactivity in multi-step organic syntheses.

Specifications

Molecular FormulaC6H12ClNO4
Molecular Weight197.62 g/mol
CAS Number14358-33-9
AppearanceWhite or Off-white Solid
Purity≥98% (by HPLC)
Melting Point115–116.5 °C (from ethanol/ethyl acetate)
Boiling Point223 °C at 760 mmHg
Flash Point88.9 °C

Industrial Applications

This aspartic acid derivative serves primarily as a chiral synthon in advanced organic synthesis, particularly in the construction of peptidomimetics and neuroactive compounds. Its protected functional groups allow for selective deprotection strategies, making it invaluable in solid-phase peptide synthesis (SPPS) and medicinal chemistry workflows.

  • Used as a building block for custom peptide sequences requiring aspartate incorporation
  • Facilitates stereoselective synthesis in API development
  • Suitable for research and large-scale GMP-compliant manufacturing

Handling and Storage

Store H-DL-Asp(OMe)-OMe hydrochloride at 2–8 °C in a tightly sealed container under dry, inert conditions. Protect from moisture and light to maintain chemical integrity. Standard packaging is 25 kg per drum, with customized options available upon request.