Intermediates

N-Boc-O-Benzyl-D-serine

  • CAS No.47173-80-8
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity N-Boc-O-Benzyl-D-serine (CAS 47173-80-8) is a key chiral building block for peptide synthesis and advanced pharmaceutical intermediates.

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Product Technical Details

Product Overview

N-Boc-O-Benzyl-D-serine is a protected D-serine derivative widely employed in the synthesis of complex peptides and bioactive molecules. Featuring both tert-butoxycarbonyl (Boc) and benzyl (Bzl) protecting groups, this compound offers excellent stability and selective deprotection capabilities, making it indispensable in solid-phase and solution-phase peptide chemistry. With a molecular formula of C15H21NO5 and a molecular weight of 295.33 g/mol, it ensures high reactivity and compatibility with standard coupling protocols.

Specifications

CAS Number47173-80-8
Molecular FormulaC15H21NO5
Molecular Weight295.33 g/mol
AppearanceWhite crystalline powder
Purity≥98% (by HPLC)
Melting Point58–60 °C (lit.)
Density1.174 g/cm³
Boiling Point456.2 °C at 760 mmHg
Flash Point229.7 °C
Refractive Index1.523

Industrial Applications

This chiral amino acid derivative serves primarily as a critical intermediate in the production of therapeutic peptides, protease inhibitors, and other high-value active pharmaceutical ingredients (APIs). Its orthogonal protection strategy enables precise control during multi-step syntheses, particularly in the development of neurological therapeutics and advanced organic synthesis pathways. It is not intended for direct human or veterinary use but is strictly for research and industrial-scale manufacturing under GMP-compliant environments.

  • Essential building block for stereoselective peptide synthesis
  • Compatible with Fmoc/Boc SPPS (solid-phase peptide synthesis) strategies
  • Enables selective deprotection for sequential coupling reactions
  • Supplied with full analytical documentation including COA and HPLC chromatograms

Stored at 2–8 °C in a tightly sealed container under dry, cool conditions to maintain integrity and extend shelf life. Packaging is available in 25 kg drums or customized configurations upon request.