Intermediates

N-Hydroxy-5-norbornene-2,3-dicarboximide

  • CAS No.21715-90-2
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity N-Hydroxy-5-norbornene-2,3-dicarboximide (CAS 21715-90-2), a specialized condensation reagent for advanced organic synthesis.

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Product Technical Details

Product Overview

N-Hydroxy-5-norbornene-2,3-dicarboximide (HONB) is a high-value bicyclic imide derivative widely employed as a condensation reagent in complex organic synthesis. With its rigid norbornene scaffold and activated N–OH functionality, HONB facilitates efficient amide and ester bond formation under mild conditions, making it particularly valuable in the preparation of sensitive intermediates for pharmaceuticals and fine chemicals.

Specifications

Molecular FormulaC9H9NO3
Molecular Weight179.17 g/mol
CAS Number21715-90-2
AppearanceOff-white to white crystalline powder
Purity (HPLC)≥99.0%
Melting Point165–170°C
Density1.574 g/cm³
Boiling Point347.7°C
Refractive Index1.673
HS Code2925190090
UN NumberUN3077
Hazard ClassClass 9
Packing GroupIII

Industrial Applications

This compound serves primarily as a coupling agent in peptide synthesis and other carboxyl activation protocols. Its structural rigidity enhances selectivity and reduces racemization, which is critical in the production of chiral active pharmaceutical ingredients (APIs). Key advantages include:

  • High reactivity with minimal side reactions
  • Compatibility with standard solid-phase and solution-phase synthesis workflows
  • Stability under ambient storage conditions when properly handled

Stored in a cool, well-ventilated area away from moisture and oxidizing agents, N-Hydroxy-5-norbornene-2,3-dicarboximide maintains integrity over extended periods. Standard packaging is 25 kg per drum, with custom options available for industrial-scale procurement.