Tianeptine
- CAS No.66981-73-5
- GradeIndustrial / Pharmaceutical
- Availability● In Stock
High-purity Tianeptine (CAS 66981-73-5), a tricyclic pharmaceutical intermediate used in advanced neurological therapeutics research and development.
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Product Overview
Tianeptine is a high-value tricyclic compound primarily utilized as a pharmaceutical intermediate in the development of advanced neurological therapeutics. With the molecular formula C21H25ClN2O4S and a molecular weight of 436.95 g/mol, it exhibits distinct pharmacological properties that differentiate it from classical tricyclic antidepressants. This product is supplied with stringent quality control to meet international standards for research and industrial-scale synthesis.
Specifications
| Molecular Formula | C21H25ClN2O4S |
|---|---|
| Molecular Weight | 436.952 g/mol |
| Exact Mass | 436.122345 |
| Melting Point | 129–131°C |
| Density | 1.4 ± 0.1 g/cm³ |
| Boiling Point | 609.2 ± 65.0 °C at 760 mmHg |
| Flash Point | 322.2 ± 34.3 °C |
| LogP | 2.57 |
| PSA | 95.09 Ų |
| Vapour Pressure | 0.0 ± 1.8 mmHg at 25°C |
| Refractive Index | 1.639 |
Quality Control
- Assay: ≥99.0%
- Residue on ignition: ≤0.20%
- Loss on drying: ≤1.0%
- Heavy metals: ≤20 ppm
- Individual impurity: ≤0.1%
- Total impurities: ≤0.5%
Industrial Applications
As a specialized intermediate, Tianeptine serves as a critical building block in the synthesis of complex pharmaceutical APIs targeting central nervous system disorders. Its unique mechanism—potentially involving modulation of glutamatergic pathways and neurotrophic factors—makes it a subject of interest in medicinal chemistry research. It is strictly intended for laboratory and industrial R&D use under compliant regulatory frameworks. This compound is not approved for direct human consumption in many jurisdictions, including the U.S., Canada, and the U.K.
Storage conditions require a cool, dry, and well-ventilated environment with the container tightly sealed to maintain stability and purity. Standard packaging is 25 kg per drum, with custom configurations available upon request.
