Intermediates

2-Amino-5-bromothiazole Monohydrobromide

  • CAS No.61296-22-8
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 2-Amino-5-bromothiazole monohydrobromide (CAS 61296-22-8), a key halogenated heterocyclic intermediate for advanced pharmaceutical and agrochemical synthesis.

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Product Technical Details

Product Overview

2-Amino-5-bromothiazole monohydrobromide is a halogenated thiazole derivative widely employed as a critical building block in the synthesis of complex pharmaceutical active ingredients and specialty agrochemicals. With its reactive bromo and amino functionalities on a rigid thiazole scaffold, this compound enables selective cross-coupling and nucleophilic substitution reactions, making it indispensable in modern medicinal chemistry workflows.

Specifications

Molecular FormulaC₃H₄Br₂N₂S
Molecular Weight259.95 g/mol
AppearanceLight yellow to light brown crystalline powder
Melting Point165 °C (dec.)
Boiling Point192.5 °C at 760 mmHg
Flash Point70.2 °C
Purity (HPLC)≥96.0% (Typical: 96.7%)

Industrial Applications

This high-purity intermediate is primarily utilized in the development of novel therapeutic agents targeting metabolic and inflammatory pathways. Its structural motif serves as a versatile precursor in Suzuki, Buchwald-Hartwig, and other palladium-catalyzed transformations. Additionally, it finds application in the synthesis of fungicides and herbicides requiring halogenated nitrogen heterocycles for optimal bioactivity.

  • Enables regioselective functionalization via bromine displacement
  • Compatible with standard peptide and small-molecule coupling protocols
  • Supplied with full analytical documentation including COA and HPLC chromatograms
  • Manufactured under ISO-compliant quality systems for consistent batch-to-batch performance