Intermediates

3-Bromo-5-chloropicolinonitrile

  • CAS No.760207-83-8
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 3-Bromo-5-chloropicolinonitrile (CAS 760207-83-8), a versatile pyridine-based building block for advanced organic synthesis in pharmaceutical and agrochemical R&D.

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Product Technical Details

Product Overview

3-Bromo-5-chloropicolinonitrile is a high-value halogenated pyridine derivative widely employed as a key intermediate in the synthesis of complex active pharmaceutical ingredients (APIs) and specialty agrochemical compounds. With its dual functional handles—bromine for cross-coupling reactions and nitrile for further derivatization—this compound offers exceptional versatility in multi-step synthetic pathways.

Specifications

Molecular FormulaC6H2BrClN2
Molecular Weight217.451 g/mol
Density1.9 ± 0.1 g/cm³
Boiling Point297.5 ± 40.0 °C at 760 mmHg
Flash Point133.7 ± 27.3 °C
AppearancePale yellow solid
Assay≥99.0%

Industrial Applications

This compound serves primarily as a critical synthon in medicinal chemistry and crop protection research. Its structural features enable efficient construction of heterocyclic scaffolds through palladium-catalyzed Suzuki, Sonogashira, or Buchwald-Hartwig reactions. Common downstream applications include the development of kinase inhibitors, antimicrobial agents, and novel herbicidal molecules.

  • Ideal for late-stage functionalization due to orthogonal reactivity of Br and CN groups
  • Compatible with standard anhydrous and inert-atmosphere reaction conditions
  • Supplied with comprehensive analytical documentation including NMR, HPLC, and MS data

Stored in a cool, well-ventilated area away from moisture and oxidizing agents, 3-Bromo-5-chloropicolinonitrile maintains stability under recommended conditions. Packaging is typically 25 kg per drum, with custom options available for large-scale industrial procurement.