Intermediates

N-Benzyloxycarbonyl-L-alaninol

  • CAS No.66674-16-6
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity N-Benzyloxycarbonyl-L-alaninol (≥98%) for use as a chiral building block in advanced pharmaceutical synthesis.

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Product Technical Details

Product Overview

N-Benzyloxycarbonyl-L-alaninol is a high-value chiral amino alcohol derivative widely employed as a protected intermediate in the synthesis of complex bioactive molecules. Featuring the benzyloxycarbonyl (Cbz or Z) protecting group on the amine and a free hydroxyl functionality, this compound offers excellent regioselectivity and stability under standard organic transformation conditions. Its stereochemical integrity makes it particularly valuable in asymmetric synthesis and the construction of peptidomimetics.

Specifications

Molecular FormulaC₁₁H₁₅NO₃
Molecular Weight209.24 g/mol
CAS Number66674-16-6
AppearanceWhite powder
Purity≥98% (by HPLC)
Moisture Content0.25%
Total Impurities0.30%
Melting Point81–84 °C (lit.)
Density1.15 g/cm³
Boiling Point375.18 °C at 760 mmHg
Refractive Index1.534
Flash Point180.70 °C

Industrial Applications

This compound serves primarily as a specialized intermediate in the pharmaceutical and fine chemical industries. Key applications include:

  • Synthesis of protease inhibitors and other enzyme-targeted therapeutics
  • Chiral auxiliary in asymmetric catalysis
  • Building block for modified peptides and peptidomimetic scaffolds
  • Precursor in the preparation of β-amino alcohols with defined stereochemistry

Due to its well-defined stereochemistry and orthogonal protecting group strategy, N-Benzyloxycarbonyl-L-alaninol enables precise molecular construction in multi-step syntheses requiring high enantiomeric fidelity.

Handling and Storage

Store at 0–5 °C in a tightly sealed container under inert atmosphere if possible. Keep in a cool, dry place away from moisture and oxidizing agents. Shelf life is typically 24 months when stored under recommended conditions. Packaging is available in 25 kg fiber drums or customized configurations upon request.