Intermediates

3-(Trifluoromethoxy)benzonitrile

  • CAS No.52771-22-9
  • GradeIndustrial / Pharmaceutical
  • Availability● In Stock

High-purity 3-(Trifluoromethoxy)benzonitrile (CAS 52771-22-9), a versatile fluorinated aromatic intermediate for advanced organic synthesis in pharmaceutical and agrochemical R&D.

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Product Technical Details

Product Overview

3-(Trifluoromethoxy)benzonitrile is a high-value fluorinated aromatic building block widely employed as a key intermediate in the synthesis of complex organic molecules. With its electron-withdrawing trifluoromethoxy and nitrile functional groups positioned meta to each other on the benzene ring, this compound offers unique reactivity and stability profiles essential for constructing bioactive scaffolds in medicinal chemistry and crop protection agents.

Specifications

Molecular FormulaC8H4F3NO
Molecular Weight187.119 g/mol
CAS Number52771-22-9
AppearanceColorless to almost colorless clear liquid
Assay≥98.0%
Density1.3 ± 0.1 g/cm³
Boiling Point178.1 ± 40.0 °C at 760 mmHg
Flash Point61.5 ± 27.3 °C
Vapor Pressure1.0 ± 0.3 mmHg at 25°C
Refractive Index1.461

Industrial Applications

This fluorinated benzonitrile derivative serves primarily as a specialty intermediate in multi-step synthetic routes. Its applications include:

  • Construction of heterocyclic cores in pharmaceutical active pharmaceutical ingredient (API) development
  • Synthesis of novel agrochemical compounds requiring enhanced metabolic stability
  • Preparation of liquid crystals and electronic materials leveraging its rigid aromatic structure
  • Use in cross-coupling reactions (e.g., Suzuki, Sonogashira) due to the robustness of the C–CN bond

Stored in a cool, well-ventilated area away from oxidizing agents, 3-(Trifluoromethoxy)benzonitrile is typically supplied in 200 kg drums or customized packaging to meet industrial-scale manufacturing demands. As a non-terminal, non-formulation chemical, it supports upstream synthesis rather than direct end-product formulation.